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Target
Cannabinoid receptor 2
Ligand
BDBM50092585
Substrate
n/a
Meas. Tech.
ChEMBL_46990 (CHEMBL658959)
Ki
113±n/a nM
Citation
 Mahadevan, A; Siegel, C; Martin, BR; Abood, ME; Beletskaya, I; Razdan, RK Novel cannabinol probes for CB1 and CB2 cannabinoid receptors. J Med Chem 43:3778-85 (2000) [PubMed]  Article 
Target
Name:
Cannabinoid receptor 2
Synonyms:
CANNABINOID CB2 | CB-2 | CB2 | CB2A | CB2B | CNR2 | CNR2_HUMAN | CX5 | Cannabinoid CB2 receptor | Cannabinoid receptor 2 (CB2) | Cannabinoid receptor 2 (CB2R) | hCB2
Type:
G Protein-Coupled Receptor (GPCR)
Mol. Mass.:
39690.94
Organism:
Homo sapiens (Human)
Description:
P34972
Residue:
360
Sequence:
MEECWVTEIANGSKDGLDSNPMKDYMILSGPQKTAVAVLCTLLGLLSALENVAVLYLILSSHQLRRKPSYLFIGSLAGADFLASVVFACSFVNFHVFHGVDSKAVFLLKIGSVTMTFTASVGSLLLTAIDRYLCLRYPPSYKALLTRGRALVTLGIMWVLSALVSYLPLMGWTCCPRPCSELFPLIPNDYLLSWLLFIAFLFSGIIYTYGHVLWKAHQHVASLSGHQDRQVPGMARMRLDVRLAKTLGLVLAVLLICWFPVLALMAHSLATTLSDQVKKAFAFCSMLCLINSMVNPVIYALRSGEIRSSAHHCLAHWKKCVRGLGSEAKEEAPRSSVTETEADGKITPWPDSRDLDLSDC
  
Inhibitor
Name:
BDBM50092585
Synonyms:
4-(1,1-Dimethyl-butyl)-2'-isopropyl-5'-methyl-biphenyl-2-ol | CHEMBL125010
Type:
Small organic molecule
Emp. Form.:
C22H30O
Mol. Mass.:
310.473
SMILES:
CCCC(C)(C)c1ccc(c(O)c1)-c1cc(C)ccc1C(C)C
Structure:
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