Reaction Details Report a problem with these data
Target
Cannabinoid receptor 2
Ligand
BDBM50092584
Substrate
n/a
Meas. Tech.
ChEMBL_46990 (CHEMBL658959)
Ki
1±n/a nM
Citation
 Mahadevan, A; Siegel, C; Martin, BR; Abood, ME; Beletskaya, I; Razdan, RK Novel cannabinol probes for CB1 and CB2 cannabinoid receptors. J Med Chem 43:3778-85 (2000) [PubMed]  Article 
Target
Name:
Cannabinoid receptor 2
Synonyms:
CANNABINOID CB2 | CB-2 | CB2 | CB2A | CB2B | CNR2 | CNR2_HUMAN | CX5 | Cannabinoid CB2 receptor | Cannabinoid receptor 2 (CB2) | Cannabinoid receptor 2 (CB2R) | hCB2
Type:
G Protein-Coupled Receptor (GPCR)
Mol. Mass.:
39690.94
Organism:
Homo sapiens (Human)
Description:
P34972
Residue:
360
Sequence:
MEECWVTEIANGSKDGLDSNPMKDYMILSGPQKTAVAVLCTLLGLLSALENVAVLYLILSSHQLRRKPSYLFIGSLAGADFLASVVFACSFVNFHVFHGVDSKAVFLLKIGSVTMTFTASVGSLLLTAIDRYLCLRYPPSYKALLTRGRALVTLGIMWVLSALVSYLPLMGWTCCPRPCSELFPLIPNDYLLSWLLFIAFLFSGIIYTYGHVLWKAHQHVASLSGHQDRQVPGMARMRLDVRLAKTLGLVLAVLLICWFPVLALMAHSLATTLSDQVKKAFAFCSMLCLINSMVNPVIYALRSGEIRSSAHHCLAHWKKCVRGLGSEAKEEAPRSSVTETEADGKITPWPDSRDLDLSDC
  
Inhibitor
Name:
BDBM50092584
Synonyms:
CHEMBL331838 | [3-(1,1-Dimethyl-heptyl)-6,6-dimethyl-6H-benzo[c]chromen-9-yl]-methanol
Type:
Small organic molecule
Emp. Form.:
C25H34O2
Mol. Mass.:
366.5363
SMILES:
CCCCCCC(C)(C)c1ccc-2c(OC(C)(C)c3ccc(CO)cc-23)c1
Structure:
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