Reaction Details Report a problem with these data
Target
Free fatty acid receptor 4
Ligand
BDBM50543523
Substrate
n/a
Meas. Tech.
ChEMBL_1989317 (CHEMBL4623052)
EC50
220±n/a nM
Citation
 Dowarah, J; Singh, VP Anti-diabetic drugs recent approaches and advancements. Bioorg Med Chem 28:0 (2020) [PubMed]  Article 
Target
Name:
Free fatty acid receptor 4
Synonyms:
FFAR4 | FFAR4_HUMAN | G-protein coupled receptor 120 | G-protein coupled receptor 129 | G-protein coupled receptor GT01 | G-protein coupled receptor PGR4 | GPR120 | GPR129 | O3FAR1 | Omega-3 fatty acid receptor 1 | PGR4 | Synonyms=GPR120
Type:
PROTEIN
Mol. Mass.:
40511.04
Organism:
Homo sapiens
Description:
ChEMBL_100956
Residue:
361
Sequence:
MSPECARAAGDAPLRSLEQANRTRFPFFSDVKGDHRLVLAAVETTVLVLIFAVSLLGNVCALVLVARRRRRGATACLVLNLFCADLLFISAIPLVLAVRWTEAWLLGPVACHLLFYVMTLSGSVTILTLAAVSLERMVCIVHLQRGVRGPGRRARAVLLALIWGYSAVAALPLCVFFRVVPQRLPGADQEISICTLIWPTIPGEISWDVSFVTLNFLVPGLVIVISYSKILQITKASRKRLTVSLAYSESHQIRVSQQDFRLFRTLFLLMVSFFIMWSPIIITILLILIQNFKQDLVIWPSLFFWVVAFTFANSALNPILYNMTLCRNEWKKIFCCFWFPEKGAILTDTSVKRNDLSIISG
  
Inhibitor
Name:
BDBM50543523
Synonyms:
CHEMBL4642294
Type:
Small organic molecule
Emp. Form.:
C24H26O4
Mol. Mass.:
378.4608
SMILES:
OC(=O)[C@H]1C[C@@H]1CCC12CCC(CC1)(O2)c1cccc(Oc2ccccc2)c1 |r|
Structure:
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