Reaction Details Report a problem with these data
Target
Free fatty acid receptor 4
Ligand
BDBM50543527
Substrate
n/a
Meas. Tech.
ChEMBL_1989316 (CHEMBL4623051)
EC50
179±n/a nM
Citation
 Dowarah, J; Singh, VP Anti-diabetic drugs recent approaches and advancements. Bioorg Med Chem 28:0 (2020) [PubMed]  Article 
Target
Name:
Free fatty acid receptor 4
Synonyms:
FFAR4 | FFAR4_HUMAN | G-protein coupled receptor 120 | G-protein coupled receptor 129 | G-protein coupled receptor GT01 | G-protein coupled receptor PGR4 | GPR120 | GPR129 | O3FAR1 | Omega-3 fatty acid receptor 1 | PGR4 | Synonyms=GPR120
Type:
PROTEIN
Mol. Mass.:
40511.04
Organism:
Homo sapiens
Description:
ChEMBL_100956
Residue:
361
Sequence:
MSPECARAAGDAPLRSLEQANRTRFPFFSDVKGDHRLVLAAVETTVLVLIFAVSLLGNVCALVLVARRRRRGATACLVLNLFCADLLFISAIPLVLAVRWTEAWLLGPVACHLLFYVMTLSGSVTILTLAAVSLERMVCIVHLQRGVRGPGRRARAVLLALIWGYSAVAALPLCVFFRVVPQRLPGADQEISICTLIWPTIPGEISWDVSFVTLNFLVPGLVIVISYSKILQITKASRKRLTVSLAYSESHQIRVSQQDFRLFRTLFLLMVSFFIMWSPIIITILLILIQNFKQDLVIWPSLFFWVVAFTFANSALNPILYNMTLCRNEWKKIFCCFWFPEKGAILTDTSVKRNDLSIISG
  
Inhibitor
Name:
BDBM50543527
Synonyms:
CHEMBL4647832
Type:
Small organic molecule
Emp. Form.:
C22H17F6NO3S
Mol. Mass.:
489.431
SMILES:
CC(Cc1cc(F)c(OCc2c(nsc2C(F)(F)F)-c2ccc(C)cc2F)c(F)c1)C(O)=O
Structure:
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