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Target
Platelet-activating factor receptor
Ligand
BDBM50118200
Substrate
n/a
Meas. Tech.
ChEMBL_155144 (CHEMBL760185)
Ki
790.0±n/a nM
Citation
 Strømgaard, K; Saito, DR; Shindou, H; Ishii, S; Shimizu, T; Nakanishi, K Ginkgolide derivatives for photolabeling studies: preparation and pharmacological evaluation. J Med Chem 45:4038-46 (2002) [PubMed]  Article 
Target
Name:
Platelet-activating factor receptor
Synonyms:
PAF-R | PTAFR_MOUSE | Platelet activating factor receptor | Platelet-activating factor receptor | Ptafr
Type:
PROTEIN
Mol. Mass.:
39163.36
Organism:
Mus musculus
Description:
ChEMBL_155144
Residue:
341
Sequence:
MEHNGSFRVDSEFRYTLFPIVYSVIFILGVVANGYVLWVFANLYPSKKLNEIKIFMVNLTMADLLFLITLPLWIVYYYNEGDWILPNFLCNVAGCLFFINTYCSVAFLGVITYNRYQAVAYPIKTAQATTRKRGISLSLIIWVSIVATASYFLATDSTNLVPNKDGSGNITRCFEHYEPYSVPILVVHVFIAFCFFLVFFLIFYCNLVIIHTLLTQPMRQQRKAGVKRRALWMVCTVLAVFIICFVPHHVVQLPWTLAELGYQTNFHQAINDAHQITLCLLSTNCVLDPVIYCFLTKKFRKHLSEKFYSMRSSRKCSRATSDTCTEVIVPANQTPIVSLKN
  
Inhibitor
Name:
BDBM50118200
Synonyms:
6-(4-azido-2,3,5,6-tetrafluorobenzyloxy)-8-(tert-butyl)-9,12,17-trihydroxy-16-methyl-2,4,14,19-tetraoxahexacyclo[8.7.2.01,11.03,7.07,11.013,17]nonadecane-5,15,18-trione | CHEMBL131402
Type:
Small organic molecule
Emp. Form.:
C27H25F4N3O11
Mol. Mass.:
643.4945
SMILES:
C[C@@H]1C(=O)O[C@H]2[C@H](O)[C@]34C5OC(=O)C3(OC3OC(=O)[C@H](OCc6c(F)c(F)c(N=[N+]=[N-])c(F)c6F)C43[C@@H]([C@H]5O)C(C)(C)C)[C@@]12O
Structure:
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