Target
Mu-type opioid receptor
Ligand
BDBM50137992
Substrate
n/a
Meas. Tech.
ChEMBL_145149 (CHEMBL755953)
Ki
90±n/a nM
Citation
 Zhang, AXiong, WBidlack, JMHilbert, JEKnapp, BIWentland, MPNeumeyer, JL 10-Ketomorphinan and 3-substituted-3-desoxymorphinan analogues as mixed kappa and micro opioid ligands: synthesis and biological evaluation of their binding affinity at opioid receptors. J Med Chem 47:165-74 (2003) [PubMed]  Article 
Target
Name:
Mu-type opioid receptor
Synonyms:
M-OR-1 | MOR-1 | Mu opioid receptor | Mu-type opioid receptor (Mu) | OPIATE Mu | OPRM1 | OPRM_CAVPO
Type:
Enzyme Catalytic Domain
Mol. Mass.:
11165.58
Organism:
GUINEA PIG
Description:
P97266
Residue:
98
Sequence:
YTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSIFTLCTMSVDRYIAVCHPVKALDFRTPRNAKTVNVCNWI
  
Inhibitor
Name:
BDBM50137992
Synonyms:
3-Hydroxy-10-keto-N-(2-methoxyethyl)morphinan | CHEMBL432873
Type:
Small organic molecule
Emp. Form.:
C19H25NO3
Mol. Mass.:
315.4067
SMILES:
COCCN1CC[C@]23CCCC[C@H]2[C@H]1C(=O)c1ccc(O)cc31
Structure:
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