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TargetLysophosphatidic acid receptor 3 (LPAR3)
LigandBDBM50150008
Substrate/Competitorn/a
Meas. Tech.ChEMBL_304755
Ki 150±n/a nM
Citation Heasley, BHJarosz, RCarter, KMVan, SJLynch, KRMacdonald, TL A novel series of 2-pyridyl-containing compounds as lysophosphatidic acid receptor antagonists: development of a nonhydrolyzable LPA3 receptor-selective antagonist. Bioorg Med Chem Lett14:4069-74 (2004) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Lysophosphatidic acid receptor 3 (LPAR3)
Name:Lysophosphatidic acid receptor 1/3
Synonyms:Lysophosphatidic acid receptor Edg-7
Type:Enzyme
Mol. Mass.:40149.72
Organism:Homo sapiens (Human)
Description:Q9UBY5
Residue:353
Sequence:
MNECHYDKHMDFFYNRSNTDTVDDWTGTKLVIVLCVGTFFCLFIFFSNSLVIAAVIKNRK
FHFPFYYLLANLAAADFFAGIAYVFLMFNTGPVSKTLTVNRWFLRQGLLDSSLTASLTNL
LVIAVERHMSIMRMRVHSNLTKKRVTLLILLVWAIAIFMGAVPTLGWNCLCNISACSSLA
PIYSRSYLVFWTVSNLMAFLIMVVVYLRIYVYVKRKTNVLSPHTSGSISRRRTPMKLMKT
VMTVLGAFVVCWTPGLVVLLLDGLNCRQCGVQHVKRWFLLLALLNSVVNPIIYSYKDEDM
YGTMKKMICCFSQENPERRPSRIPSTVLSRSDTGSQYIEDSISQGAVCNKSTS
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM50150008
NameBDBM50150008
Synonyms:CHEMBL182773 | [4-[4-(4-Methoxy-3,5-dimethyl-pyridin-2-ylmethoxy)-phenyl]-3-((Z)-(R)-octadec-9-enoylamino)-butyl]-phosphonic acid
TypeSmall organic molecule
Emp. Form.C37H59N2O6P
Mol. Mass.658.8479
SMILESCCCCCCCC\C=C/CCCCCCCC(=O)N[C@@H](CCP(O)(O)=O)Cc1ccc(OCc2ncc(C)c(OC)c2C)cc1
Structure
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n/a