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TargetLysophosphatidic acid receptor 3 (LPAR3)
LigandBDBM50176392
Substrate/Competitorn/a
Meas. Tech.ChEMBL_333864
Ki 118±n/a nM
Citation Durgam, GGTsukahara, RMakarova, NWalker, MDFujiwara, YPigg, KRBaker, DLSardar, VMParrill, ALTigyi, GMiller, DD Synthesis and pharmacological evaluation of second-generation phosphatidic acid derivatives as lysophosphatidic acid receptor ligands. Bioorg Med Chem Lett16:633-40 (2005) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Lysophosphatidic acid receptor 3 (LPAR3)
Name:Lysophosphatidic acid receptor 1/3
Synonyms:Lysophosphatidic acid receptor Edg-7
Type:Enzyme
Mol. Mass.:40149.72
Organism:Homo sapiens (Human)
Description:Q9UBY5
Residue:353
Sequence:
MNECHYDKHMDFFYNRSNTDTVDDWTGTKLVIVLCVGTFFCLFIFFSNSLVIAAVIKNRK
FHFPFYYLLANLAAADFFAGIAYVFLMFNTGPVSKTLTVNRWFLRQGLLDSSLTASLTNL
LVIAVERHMSIMRMRVHSNLTKKRVTLLILLVWAIAIFMGAVPTLGWNCLCNISACSSLA
PIYSRSYLVFWTVSNLMAFLIMVVVYLRIYVYVKRKTNVLSPHTSGSISRRRTPMKLMKT
VMTVLGAFVVCWTPGLVVLLLDGLNCRQCGVQHVKRWFLLLALLNSVVNPIIYSYKDEDM
YGTMKKMICCFSQENPERRPSRIPSTVLSRSDTGSQYIEDSISQGAVCNKSTS
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  Blast E-value cutoff:
BDBM50176392
NameBDBM50176392
Synonyms:CHEMBL379248 | thiophosphoric acid (R)-2-octanoylamino-2-octylcarbamoyl-ethyl ester
TypeSmall organic molecule
Emp. Form.C19H39N2O5PS
Mol. Mass.438.562
SMILESCCCCCCCCNC(=O)[C@@H](COP(O)(O)=S)NC(=O)CCCCCCC
Structure
Search PDB for entries with ligand similarity:Similarity to this molecule at least:
n/a