Reaction Details Report a problem with these data
Target
Phospholipase A2
Ligand
BDBM50262842
Substrate
n/a
Meas. Tech.
ChEMBL_489269 (CHEMBL990825)
IC50
950±n/a nM
Citation
Oslund, RC; Cermak, N; Gelb, MH Highly specific and broadly potent inhibitors of mammalian secreted phospholipases A2. J Med Chem 51:4708-14 (2008) [PubMed] Article
More Info.:
Target
Name:
Phospholipase A2
Synonyms:
PA21B_MOUSE | Phospholipase A2 group 1B | Pla2 | Pla2g1b
Type:
PROTEIN
Mol. Mass.:
16291.94
Organism:
Mus musculus
Description:
ChEMBL_489269
Residue:
146
Sequence:
MKLLLLAALLTAGAAAHSISPRAVWQFRNMIKCTIPGSDPLKDYNNYGCYCGLGGWGTPVDDLDRCCQTHDHCYSQAKKLESCKFLIDNPYTNTYSYSCSGSEITCSAKNNKCEDFICNCDREAAICFSKVPYNKEYKNLDTGKFC