Reaction Details Report a problem with these data
Target
Group 10 secretory phospholipase A2
Ligand
BDBM50263001
Substrate
n/a
Meas. Tech.
ChEMBL_489281 (CHEMBL990837)
IC50
>1600±n/a nM
Citation
Oslund, RC; Cermak, N; Gelb, MH Highly specific and broadly potent inhibitors of mammalian secreted phospholipases A2. J Med Chem 51:4708-14 (2008) [PubMed] Article
More Info.:
Target
Name:
Group 10 secretory phospholipase A2
Synonyms:
Group X secretory phospholipase A2 | PA2GX_MOUSE | Pla2g10
Type:
PROTEIN
Mol. Mass.:
17005.09
Organism:
Mus musculus
Description:
ChEMBL_537139
Residue:
151
Sequence:
MLLLLLLLLLGPGPGFSEATRRSHVYKRGLLELAGTLDCVGPRSPMAYMNYGCYCGLGGHGEPRDAIDWCCYHHDCCYSRAQDAGCSPKLDRYPWKCMDHHILCGPAENKCQELLCRCDEELAYCLAGTEYHLKYLFFPSILCEKDSPKCN