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Target
Phospholipase A2 group V
Ligand
BDBM50274391
Substrate
n/a
Meas. Tech.
ChEMBL_537133 (CHEMBL989793)
IC50
>1600±n/a nM
Citation
 Oslund, RC; Cermak, N; Verlinde, CL; Gelb, MH Simplified YM-26734 inhibitors of secreted phospholipase A2 group IIA. Bioorg Med Chem Lett 18:5415-9 (2008) [PubMed]  Article 
Target
Name:
Phospholipase A2 group V
Synonyms:
PA2G5_MOUSE | Pla2g5
Type:
PROTEIN
Mol. Mass.:
15864.30
Organism:
Mus musculus
Description:
ChEMBL_700980
Residue:
137
Sequence:
MKGLLTLAWFLACSVPAVPGGLLELKSMIEKVTGKNAFKNYGFYGCYCGWGGRGTPKDGTDWCCQMHDRCYGQLEEKDCAIRTQSYDYRYTNGLVICEHDSFCPMRLCACDRKLVYCLRRNLWTYNPLYQYYPNFLC
  
Inhibitor
Name:
BDBM50274391
Synonyms:
1-(3-dodecyl-2,4,6-trihydroxyphenyl)dodecan-1-one | CHEMBL483761
Type:
Small organic molecule
Emp. Form.:
C30H52O4
Mol. Mass.:
476.7315
SMILES:
CCCCCCCCCCCCc1c(O)cc(O)c(C(=O)CCCCCCCCCCC)c1O
Structure:
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