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TargetCalcitonin gene-related peptide (CGRP alpha)
LigandBDBM50246709
Substrate/Competitorn/a
Meas. Tech.ChEMBL_556924
IC50 0.790000±n/a nM
Citation Miranda, LPHolder, JRShi, LBennett, BAral, JGegg, CVWright, MWalker, KDoellgast, GRogers, RLi, HValladares, VSalyers, KJohnson, EWild, K Identification of potent, selective, and metabolically stable peptide antagonists to the calcitonin gene-related peptide (CGRP) receptor. J Med Chem51:7889-97 (2008) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Calcitonin gene-related peptide (CGRP alpha)
Name:Calcitonin gene-related peptide (CGRP alpha)
Synonyms:CGRP | Calcitonin gene-related peptide 1
Type:Enzyme
Mol. Mass.:13902.80
Organism:Homo sapiens (Human)
Description:P06881
Residue:128
Sequence:
MGFQKFSPFLALSILVLLQAGSLHAAPFRSALESSPADPATLSEDEARLLLAALVQNYVQ
MKASELEQEQEREGSRIIAQKRACDTATCVTHRLAGLLSRSGGVVKNNFVPTNVGSKAFG
RRRRDLQA
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BDBM50246709
NameBDBM50246709
Synonyms:Ac-WVTH[Cit]LAGLLS[Cit]SGGVV[hArg]KNFVPTDVGP[2-Nal]AF-NH2 | CHEMBL509603
TypeSmall organic molecule
Emp. Form.C164H248N44O41
Mol. Mass.3491.9941
SMILESn/a
Structure
Search PDB for entries with ligand similarity:Similarity to this molecule at least:
n/a