Reaction Details Report a problem with these data
Target
Chymotrypsin-like protease CTRL-1
Ligand
BDBM50288610
Substrate
n/a
Meas. Tech.
ChEBML_49606
IC50
>1000±n/a nM
Citation
Iqbal, M; Chatterjee, S; Kauer, JC; Mallamo, JP; Messina, PA; Reiboldt, A; Siman, R Potent α-ketocarbonyl and boronic ester derived inhibitors of proteasome Bioorg Med Chem Lett 6:287-290 (1996) Article
More Info.:
Target
Name:
Chymotrypsin-like protease CTRL-1
Synonyms:
CTRL | CTRL1 | CTRL_HUMAN
Type:
PROTEIN
Mol. Mass.:
28008.18
Organism:
Homo sapiens (Human)
Description:
ChEMBL_49606
Residue:
264
Sequence:
MLLLSLTLSLVLLGSSWGCGIPAIKPALSFSQRIVNGENAVLGSWPWQVSLQDSSGFHFCGGSLISQSWVVTAAHCNVSPGRHFVVLGEYDRSSNAEPLQVLSVSRAITHPSWNSTTMNNDVTLLKLASPAQYTTRISPVCLASSNEALTEGLTCVTTGWGRLSGVGNVTPAHLQQVALPLVTVNQCRQYWGSSITDSMICAGGAGASSCQGDSGGPLVCQKGNTWVLIGIVSWGTKNCNVRAPAVYTRVSKFSTWINQVIAYN