Reaction Details Report a problem with these data
Target
Calmodulin-1
Ligand
BDBM7461
Substrate
n/a
Meas. Tech.
ChEMBL_698552 (CHEMBL1647727)
IC50
33430±n/a nM
Citation
Torres-Piedra, M; Figueroa, M; Hernández-Abreu, O; Ibarra-Barajas, M; Navarrete-Vázquez, G; Estrada-Soto, S Vasorelaxant effect of flavonoids through calmodulin inhibition: Ex vivo, in vitro, and in silico approaches. Bioorg Med Chem 19:542-6 (2011) [PubMed] Article
More Info.:
Target
Name:
Calmodulin-1
Synonyms:
CALM | CALM1 | CALM1_HUMAN | CALM2 | CAM | CAM1 | CAM2 | CAMB | Calmodulin-2
Type:
Protein
Mol. Mass.:
16813.73
Organism:
Human
Description:
P0DP23
Residue:
149
Sequence:
MADQLTEEQIAEFKEAFSLFDKDGDGTITTKELGTVMRSLGQNPTEAELQDMINEVDADGNGTIDFPEFLTMMARKMKDTDSEEEIREAFRVFDKDGNGYISAAELRHVMTNLGEKLTDEEVDEMIREADIDGDGQVNYEEFVQMMTAK