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Target
cAMP-dependent protein kinase catalytic subunit PRKX
Ligand
BDBM60665
Substrate
n/a
Meas. Tech.
ChEMBL_774456 (CHEMBL1908673)
Kd
>10000±n/a nM
Citation
Davis, MI; Hunt, JP; Herrgard, S; Ciceri, P; Wodicka, LM; Pallares, G; Hocker, M; Treiber, DK; Zarrinkar, PP Comprehensive analysis of kinase inhibitor selectivity. Nat Biotechnol 29:1046-51 (2011) [PubMed] Article
More Info.:
Target
Name:
cAMP-dependent protein kinase catalytic subunit PRKX
Synonyms:
PKX1 | PRKX | PRKX_HUMAN | Serine/threonine-protein kinase PRKX
Type:
Enzyme Catalytic Domain
Mol. Mass.:
40897.91
Organism:
Homo sapiens (Human)
Description:
gi_4826948
Residue:
358
Sequence:
MEAPGLAQAAAAESDSRKVAEETPDGAPALCPSPEALSPEPPVYSLQDFDTLATVGTGTFGRVHLVKEKTAKHFFALKVMSIPDVIRLKQEQHVHNEKSVLKEVSHPFLIRLFWTWHDERFLYMLMEYVPGGELFSYLRNRGRFSSTTGLFYSAEIICAIEYLHSKEIVYRDLKPENILLDRDGHIKLTDFGFAKKLVDRTWTLCGTPEYLAPEVIQSKGHGRAVDWWALGILIFEMLSGFPPFFDDNPFGIYQKILAGKIDFPRHLDFHVKDLIKKLLVVDRTRRLGNMKNGANDVKHHRWFRSVDWEAVPQRKLKPPIVPKIAGDGDTSNFETYPENDWDTAAPVPQKDLEIFKNF