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TargetCalcitonin gene-related peptide (CGRP alpha)
LigandBDBM50356288
Substrate/Competitorn/a
Meas. Tech.ChEMBL_775006
Ki>100000±n/a nM
Citation Zartman, CBBell, IMGallicchio, SNGraham, SLKane, SAMallee, JJRutledge, RZSalvatore, CAVacca, JPWilliams, TM Identification of a novel RAMP-independent CGRP receptor antagonist. Bioorg Med Chem Lett21:6705-8 (2011) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Calcitonin gene-related peptide (CGRP alpha)
Name:Calcitonin gene-related peptide (CGRP alpha)
Synonyms:CGRP | Calcitonin gene-related peptide 1
Type:Enzyme
Mol. Mass.:13902.80
Organism:Homo sapiens (Human)
Description:P06881
Residue:128
Sequence:
MGFQKFSPFLALSILVLLQAGSLHAAPFRSALESSPADPATLSEDEARLLLAALVQNYVQ
MKASELEQEQEREGSRIIAQKRACDTATCVTHRLAGLLSRSGGVVKNNFVPTNVGSKAFG
RRRRDLQA
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BDBM50356288
NameBDBM50356288
Synonyms:CHEMBL1910942
TypeSmall organic molecule
Emp. Form.C20H19FN4O3S
Mol. Mass.414.453
SMILESFc1ccc(CNC(=O)c2cc3ncccc3c(n2)N2CCCCS2(=O)=O)cc1
Structure
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