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TargetCalcitonin gene-related peptide (CGRP alpha)
LigandBDBM50356289
Substrate/Competitorn/a
Meas. Tech.ChEMBL_775006
Ki 26000±n/a nM
Citation Zartman, CBBell, IMGallicchio, SNGraham, SLKane, SAMallee, JJRutledge, RZSalvatore, CAVacca, JPWilliams, TM Identification of a novel RAMP-independent CGRP receptor antagonist. Bioorg Med Chem Lett21:6705-8 (2011) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Calcitonin gene-related peptide (CGRP alpha)
Name:Calcitonin gene-related peptide (CGRP alpha)
Synonyms:CGRP | Calcitonin gene-related peptide 1
Type:Enzyme
Mol. Mass.:13902.80
Organism:Homo sapiens (Human)
Description:P06881
Residue:128
Sequence:
MGFQKFSPFLALSILVLLQAGSLHAAPFRSALESSPADPATLSEDEARLLLAALVQNYVQ
MKASELEQEQEREGSRIIAQKRACDTATCVTHRLAGLLSRSGGVVKNNFVPTNVGSKAFG
RRRRDLQA
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  Blast E-value cutoff:
BDBM50356289
NameBDBM50356289
Synonyms:CHEMBL1910943
TypeSmall organic molecule
Emp. Form.C21H20FN3O4S
Mol. Mass.429.465
SMILESOc1c(nc(N2CCCCS2(=O)=O)c2ccccc12)C(=O)NCc1cccc(F)c1
Structure
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