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Target
Riboflavin-binding protein
Ligand
BDBM50362897
Substrate
n/a
Meas. Tech.
ChEMBL_800332 (CHEMBL1948178)
pH
7.4±n/a
Kd
61±n/a nM
Comments
extracted
Citation
 Plantinga, A; Witte, A; Li, MH; Harmon, A; Choi, SK; Banaszak Holl, MM; Orr, BG; Baker, JR; Sinniah, K Bioanalytical Screening of Riboflavin Antagonists for Targeted Drug Delivery - A Thermodynamic and Kinetic Study. ACS Med Chem Lett 2:363-367 (2011) [PubMed]  Article 
Target
Name:
Riboflavin-binding protein
Synonyms:
RBP | RBP_CHICK | Riboflavin-binding protein, plasma form | Riboflavin-binding protein, yolk major form | Riboflavin-binding protein, yolk minor form
Type:
PROTEIN
Mol. Mass.:
27203.20
Organism:
Gallus gallus
Description:
ChEMBL_800332
Residue:
238
Sequence:
MLRFAITLFAVITSSTCQQYGCLEGDTHKANPSPEPNMHECTLYSESSCCYANFTEQLAHSPIIKVSNSYWNRCGQLSKSCEDFTKKIECFYRCSPHAARWIDPRYTAAIQSVPLCQSFCDDWYEACKDDSICAHNWLTDWERDESGENHCKSKCVPYSEMYANGTDMCQSMWGESFKVSESSCLCLQMNKKDMVAIKHLLSESSEESSSMSSSEEHACQKKLLKFEALQQEEGEERR
  
Inhibitor
Name:
BDBM50362897
Synonyms:
LUMIFLAVIN
Type:
Small organic molecule
Emp. Form.:
C13H12N4O2
Mol. Mass.:
256.26
SMILES:
Cc1cc2nc3c(nc(=O)[nH]c3=O)n(C)c2cc1C
Structure:
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