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Target
Mu-type opioid receptor
Ligand
BDBM50365855
Substrate
n/a
Meas. Tech.
ChEMBL_806704 (CHEMBL1958664)
Ki
0.08±n/a nM
Citation
Lunn, G; Roberts, LR; Content, S; Critcher, DJ; Douglas, S; Fenwick, AE; Gethin, DM; Goodwin, G; Greenway, D; Greenwood, S; Hall, K; Thomas, M; Thompson, S; Williams, D; Wood, G; Wylie, A SAR and biological evaluation of 3-azabicyclo[3.1.0]hexane derivatives asµ opioid ligands. Bioorg Med Chem Lett 22:2200-3 (2012) [PubMed] Article
More Info.:
Target
Name:
Mu-type opioid receptor
Synonyms:
M-OR-1 | MOP | MOR-1 | MOR1 | MUOR1 | Mu Opioid Receptor | Mu opiate receptor | OPIATE Mu | OPRM1 | OPRM_HUMAN | hMOP | mu-type opioid receptor isoform MOR-1
Type:
G Protein-Coupled Receptor (GPCR)
Mol. Mass.:
44789.51
Organism:
Homo sapiens (Human)
Description:
P35372
Residue:
400
Sequence:
MDSSAAPTNASNCTDALAYSSCSPAPSPGSWVNLSHLDGNLSDPCGPNRTDLGGRDSLCPPTGSPSMITAITIMALYSIVCVVGLFGNFLVMYVIVRYTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSIFTLCTMSVDRYIAVCHPVKALDFRTPRNAKIINVCNWILSSAIGLPVMFMATTKYRQGSIDCTLTFSHPTWYWENLLKICVFIFAFIMPVLIITVCYGLMILRLKSVRMLSGSKEKDRNLRRITRMVLVVVAVFIVCWTPIHIYVIIKALVTIPETTFQTVSWHFCIALGYTNSCLNPVLYAFLDENFKRCFREFCIPTSSNIEQQNSTRIRQNTRDHPSTANTVDRTNHQLENLEAETAPLP