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Target
Platelet-activating factor receptor
Ligand
BDBM50366241
Substrate
n/a
Meas. Tech.
ChEMBL_155156 (CHEMBL760196)
Ki
103±n/a nM
Citation
Sahoo, SP; Graham, DW; Acton, J; Biftu, T; Bugianesi, RL; Girotra, NN; Kuo, C; Ponpipom, MM; Doebber, TW; Wu, MS; Hwang, S; Lam, M; MacIntyre, D; Bach, TJ; Luell, S; Meurer, R; Davies, P; Alberts, AW; Chabala, JC Synthesis and biological activity of MK 287 (L-680,573): a potent, specific and orally active paf receptor antagonist Bioorg Med Chem Lett 1:327-332 (1991) Article
More Info.:
Target
Name:
Platelet-activating factor receptor
Synonyms:
PAF-R | PTAFR | PTAFR_CAVPO | Platelet activating factor receptor | Platelet-activating factor receptor
Type:
Protein
Mol. Mass.:
39005.63
Organism:
Cavia porcellus
Description:
n/a
Residue:
342
Sequence:
MELNSSSRVDSEFRYTLFPIVYSIIFVLGIIANGYVLWVFARLYPSKKLNEIKIFMVNLTVADLLFLITLPLWIVYYSNQGNWFLPKFLCNLAGCLFFINTYCSVAFLGVITYNRFQAVKYPIKTAQATTRKRGIALSLVIWVAIVAAASYFLVMDSTNVVSNKAGSGNITRCFEHYEKGSKPVLIIHICIVLGFFIVFLLILFCNLVIIHTLLRQPVKQQRNAEVRRRALWMVCTVLAVFVICFVPHHMVQLPWTLAELGMWPSSNHQAINDAHQVTLCLLSTNCVLDPVIYCFLTKKFRKHLSEKLNIMRSSQKCSRVTTDTGTEMAIPINHTPVNPIKN