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Target
Mu-type opioid receptor
Ligand
BDBM50082339
Substrate
n/a
Meas. Tech.
ChEMBL_138731 (CHEMBL747753)
Kd
4667±n/a nM
Citation
 Thomas, JB; Herault, XM; Rothman, RB; Burgess, JP; Mascarella, SW; Xu, H; Horel, RB; Dersch, CM; Carroll, FI (+/-)-4-[(N-allyl-cis-3-methyl-4-piperidinyl)phenylamino]-N,N-diethylbenzamide displays selective binding for the delta opioid receptor. Bioorg Med Chem Lett 9:3053-6 (1999) [PubMed]  Article 
Target
Name:
Mu-type opioid receptor
Synonyms:
M-OR-1 | MOR-1 | Mu opioid receptor | Mu-type opioid receptor (Mu) | OPIATE Mu | OPRM1 | OPRM_CAVPO
Type:
Enzyme Catalytic Domain
Mol. Mass.:
11165.58
Organism:
GUINEA PIG
Description:
P97266
Residue:
98
Sequence:
YTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSIFTLCTMSVDRYIAVCHPVKALDFRTPRNAKTVNVCNWI
  
Inhibitor
Name:
BDBM50082339
Synonyms:
4-[((S)-1-Allyl-3-methyl-piperidin-4-yl)-phenyl-amino]-N,N-diethyl-benzamide | CHEMBL430475
Type:
Small organic molecule
Emp. Form.:
C26H35N3O
Mol. Mass.:
405.5756
SMILES:
CCN(CC)C(=O)c1ccc(cc1)N([C@H]1CCN(CC=C)CC1C)c1ccccc1
Structure:
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