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Target
D(2) dopamine receptor
Ligand
BDBM50088756
Substrate
n/a
Meas. Tech.
ChEBML_61447
Ki
>10000±n/a nM
Citation
 Tamagnan, G; Baldwin, RM; Kula, NS; Baldessarini, RJ; Innis, RB Cyclopentadienyltricarbonylrheniumbenzazepines: synthesis and binding affinity. Bioorg Med Chem Lett 10:1113-5 (2000) [PubMed]  Article 
Target
Name:
D(2) dopamine receptor
Synonyms:
DOPAMINE D2 | DRD2_MOUSE | Dopamine D2 receptor | Dopamine Receptor D2 | Drd2
Type:
Enzyme
Mol. Mass.:
50957.64
Organism:
Mus musculus (Mouse)
Description:
P61168
Residue:
444
Sequence:
MDPLNLSWYDDDLERQNWSRPFNGSEGKPDRPHYNYYAMLLTLLIFIIVFGNVLVCMAVSREKALQTTTNYLIVSLAVADLLVATLVMPWVVYLEVVGEWKFSRIHCDIFVTLDVMMCTASILNLCAISIDRYTAVAMPMLYNTRYSSKRRVTVMIAIVWVLSFTISCPLLFGLNNTDQNECIIANPAFVVYSSIVSFYVPFIVTLLVYIKIYIVLRKRRKRVNTKRSSRAFRANLKTPLKGNCTHPEDMKLCTVIMKSNGSFPVNRRRMDAARRAQELEMEMLSSTSPPERTRYSPIPPSHHQLTLPDPSHHGLHSNPDSPAKPEKNGHAKIVNPRIAKFFEIQTMPNGKTRTSLKTMSRRKLSQQKEKKATQMLAIVLGVFIICWLPFFITHILNIHCDCNIPPVLYSAFTWLGYVNSAVNPIIYTTFNIEFRKAFMKILHC
  
Inhibitor
Name:
BDBM50088756
Synonyms:
CHEMBL427996 | Cyclopentadienyltricarbonylrheniumbenzazepine (3`-CPTR-SCH-23390)
Type:
Small organic molecule
Emp. Form.:
C26H24ClNO5Re
Mol. Mass.:
652.132
SMILES:
CN1CCc2cc(Cl)c(O)cc2C(C1)c1cccc(c1)C(=O)C1=CC=C[C@@H]1[Re](C=O)(C=O)C=O |c:27,t:25|
Structure:
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