Target
Mu-type opioid receptor
Ligand
BDBM50105498
Substrate
n/a
Meas. Tech.
ChEBML_145282
Ki
0.180000±n/a nM
Citation
 Neumeyer, JLGu, XHvan Vliet, LADeNunzio, NJRusovici, DECohen, DJNegus, SSMello, NKBidlack, JM Mixed kappa agonists and mu agonists/antagonists as potential pharmacotherapeutics for cocaine abuse: synthesis and opioid receptor binding affinity of N-substituted derivatives of morphinan. Bioorg Med Chem Lett 11:2735-40 (2001) [PubMed]  Article 
Target
Name:
Mu-type opioid receptor
Synonyms:
M-OR-1 | MOR-1 | Mu opioid receptor | Mu-type opioid receptor (Mu) | OPIATE Mu | OPRM1 | OPRM_CAVPO
Type:
Enzyme Catalytic Domain
Mol. Mass.:
11165.58
Organism:
GUINEA PIG
Description:
P97266
Residue:
98
Sequence:
YTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSIFTLCTMSVDRYIAVCHPVKALDFRTPRNAKTVNVCNWI
  
Inhibitor
Name:
BDBM50105498
Synonyms:
17-(3-fluoropropyl)-(1R,9R,10R)-17-azatetracyclo[7.5.3.01,10.02,7]heptadeca-2(7),3,5-trien-5-ol | CHEMBL419511
Type:
Small organic molecule
Emp. Form.:
C19H26FNO
Mol. Mass.:
303.4142
SMILES:
Oc1ccc2c(C[C@@H]3[C@@H]4CCCCC24CCN3CCCF)c1 |THB:17:16:8:4.5.6|
Structure:
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