Reaction Details Report a problem with these data
Target
Melanocortin receptor 5
Ligand
BDBM50129191
Substrate
n/a
Meas. Tech.
ChEBML_106667
EC50
30500±n/a nM
Citation
 Joseph, CG; Bauzo, RM; Xiang, Z; Haskell-Luevano, C Urea small molecule agonists on mouse melanocortin receptors. Bioorg Med Chem Lett 13:2079-82 (2003) [PubMed]  Article 
Target
Name:
Melanocortin receptor 5
Synonyms:
MC5R_MOUSE | Mc5r | Melanocortin receptor 5 | Melanocortin receptor 5 (MC5R)
Type:
Enzyme
Mol. Mass.:
36966.58
Organism:
Mus musculus (Mouse)
Description:
P41149
Residue:
325
Sequence:
MNSSSTLTVLNLTLNASEDGILGSNVKNKSLACEEMGIAVEVFLTLGLVSLLENILVIGAIVKNKNLHSPMYFFVGSLAVADMLVSMSNAWETVTIYLLNNKHLVIADTFVRHIDNVFDSMICISVVASMCSLLAIAVDRYITIFYALRYHHIMTARRSGVIIACIWTFCISCGIVFIIYYESKYVIICLISMFFTMLFFMVSLYIHMFLLARNHVKRIAASPRYNSVRQRTSMKGAITLTMLLGIFIVCWSPFFLHLILMISCPQNVYCSCFMSYFNMYLILIMCNSVIDPLIYALRSQEMRRTFKEIVCCHGFRRPCRLLGGY
  
Inhibitor
Name:
BDBM50129191
Synonyms:
CHEMBL305559 | N-(4-Amino-butyl)-2-(3-benzyl-ureido)-3-(1H-indol-3-yl)-propionamide
Type:
Small organic molecule
Emp. Form.:
C23H29N5O2
Mol. Mass.:
407.5087
SMILES:
NCCCCNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)NCc1ccccc1
Structure:
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