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TargetSigma non-opioid intracellular receptor 1
LigandBDBM50041245
Substrate/Competitorn/a
Meas. Tech.ChEBML_201295
Ki 4.8±n/a nM
Citation Glennon, RASmith, JDIsmaiel, AMel-Ashmawy, MBattaglia, GFischer, JB Identification and exploitation of the sigma-opiate pharmacophore. J Med Chem34:1094-8 (1991) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Sigma non-opioid intracellular receptor 1
Name:Sigma non-opioid intracellular receptor 1
Synonyms:Opioid receptor | Sigma | Sigma opioid receptor | Sigma-1
Type:Enzyme Catalytic Domain
Mol. Mass.:25266.54
Organism:RAT
Description:Q9R0C9
Residue:223
Sequence:
MPWAVGRRWAWITLFLTIVAVLIQAVWLWLGTQSFVFQREEIAQLARQYAGLDHELAFSR
LIVELRRLHPGHVLPDEELQWVFVNAGGWMGAMCLLHASLSEYVLLFGTALGSHGHSGRY
WAEISDTIISGTFHQWREGTTKSEVYYPGETVVHGPGEATAVEWGPNTWMVEYGRGVIPS
TLAFALSDTIFSTQDFLTLFYTLRAYARGLRLELTTYLFGQDP
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM50041245
NameBDBM50041245
Synonyms:((S)-1-Methyl-2-phenyl-ethyl)-phenethyl-amine | CHEMBL20804
TypeSmall organic molecule
Emp. Form.C17H21N
Mol. Mass.239.3553
SMILESC[C@@H](Cc1ccccc1)NCCc1ccccc1
Structure
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n/a