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Target
Mu-type opioid receptor
Ligand
BDBM50000785
Substrate
n/a
Meas. Tech.
ChEBML_146255
Ki
13000±n/a nM
Citation
 Cheng, CY; Wu, SC; Hsin, LW; Tam, SW Selective reversible and irreversible ligands for the kappa opioid receptor. J Med Chem 35:2243-7 (1992) [PubMed]  Article 
Target
Name:
Mu-type opioid receptor
Synonyms:
M-OR-1 | MOR-1 | Mu opioid receptor | Mu-type opioid receptor (Mu) | OPIATE Mu | OPRM1 | OPRM_CAVPO
Type:
Enzyme Catalytic Domain
Mol. Mass.:
11165.58
Organism:
GUINEA PIG
Description:
P97266
Residue:
98
Sequence:
YTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSIFTLCTMSVDRYIAVCHPVKALDFRTPRNAKTVNVCNWI
  
Inhibitor
Name:
BDBM50000785
Synonyms:
2-(3,4-Dichloro-phenyl)-N-methyl-N-(5-oxo-2-pyrrolidin-1-yl-cyclohexyl)-acetamide | CHEMBL74010
Type:
Small organic molecule
Emp. Form.:
C19H24Cl2N2O2
Mol. Mass.:
383.312
SMILES:
CN([C@H]1CC(=O)CC[C@@H]1N1CCCC1)C(=O)Cc1ccc(Cl)c(Cl)c1
Structure:
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