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Reaction Details
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TargetPlatelet activating factor receptor
LigandBDBM50006077
Substrate/Competitorn/a
Meas. Tech.ChEBML_221704
IC50 1210±n/a nM
Citation Wissner, ACarroll, MLGreen, KEKerwar, SSPickett, WCSchaub, RETorley, LWWrenn, SKohler, CA Analogues of platelet activating factor. 6. Mono- and bis-aryl phosphate antagonists of platelet activating factor. J Med Chem35:1650-62 (1992) [PubMed]  Article
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Platelet activating factor receptor
Name:Platelet activating factor receptor
Synonyms:PAF-R | Platelet-activating factor receptor
Type:Protein
Mol. Mass.:39005.63
Organism:Cavia porcellus
Description:n/a
Residue:342
Sequence:
MELNSSSRVDSEFRYTLFPIVYSIIFVLGIIANGYVLWVFARLYPSKKLNEIKIFMVNLT
VADLLFLITLPLWIVYYSNQGNWFLPKFLCNLAGCLFFINTYCSVAFLGVITYNRFQAVK
YPIKTAQATTRKRGIALSLVIWVAIVAAASYFLVMDSTNVVSNKAGSGNITRCFEHYEKG
SKPVLIIHICIVLGFFIVFLLILFCNLVIIHTLLRQPVKQQRNAEVRRRALWMVCTVLAV
FVICFVPHHMVQLPWTLAELGMWPSSNHQAINDAHQVTLCLLSTNCVLDPVIYCFLTKKF
RKHLSEKLNIMRSSQKCSRVTTDTGTEMAIPINHTPVNPIKN
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  Blast E-value cutoff:
BDBM50006077
NameBDBM50006077
Synonyms:3-{3-[(2-Ethyl-4-tetradecyl-phenoxy)-hydroxy-phosphoryloxy]-benzyl}-5-methyl-thiazol-3-ium | CHEMBL47219
TypeSmall organic molecule
Emp. Form.C33H48NO4PS
Mol. Mass.585.777
SMILESCCCCCCCCCCCCCCc1ccc(OP([O-])(=O)Oc2cccc(C[n+]3csc(C)c3)c2)c(CC)c1
Structure
Search PDB for entries with ligand similarity:Similarity to this molecule at least:
n/a