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Reaction Details
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TargetPlatelet activating factor receptor
LigandBDBM50006020
Substrate/Competitorn/a
Meas. Tech.ChEBML_221704
IC50 1490±n/a nM
Citation Wissner, ACarroll, MLGreen, KEKerwar, SSPickett, WCSchaub, RETorley, LWWrenn, SKohler, CA Analogues of platelet activating factor. 6. Mono- and bis-aryl phosphate antagonists of platelet activating factor. J Med Chem35:1650-62 (1992) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Platelet activating factor receptor
Name:Platelet activating factor receptor
Synonyms:PAF-R | Platelet-activating factor receptor
Type:Protein
Mol. Mass.:39005.63
Organism:Cavia porcellus
Description:n/a
Residue:342
Sequence:
MELNSSSRVDSEFRYTLFPIVYSIIFVLGIIANGYVLWVFARLYPSKKLNEIKIFMVNLT
VADLLFLITLPLWIVYYSNQGNWFLPKFLCNLAGCLFFINTYCSVAFLGVITYNRFQAVK
YPIKTAQATTRKRGIALSLVIWVAIVAAASYFLVMDSTNVVSNKAGSGNITRCFEHYEKG
SKPVLIIHICIVLGFFIVFLLILFCNLVIIHTLLRQPVKQQRNAEVRRRALWMVCTVLAV
FVICFVPHHMVQLPWTLAELGMWPSSNHQAINDAHQVTLCLLSTNCVLDPVIYCFLTKKF
RKHLSEKLNIMRSSQKCSRVTTDTGTEMAIPINHTPVNPIKN
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM50006020
NameBDBM50006020
Synonyms:1-{3-[Hydroxy-(2-methoxy-3-tetradecyloxy-phenoxy)-phosphoryloxy]-benzyl}-7aH-benzoimidazol-1-ium | CHEMBL296432
TypeSmall organic molecule
Emp. Form.C35H47N2O6P
Mol. Mass.622.7312
SMILESCCCCCCCCCCCCCCOc1cccc(OP([O-])(=O)Oc2cccc(C[n+]3c[nH]c4ccccc34)c2)c1OC
Structure
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n/a