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Reaction Details
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TargetPlatelet activating factor receptor
LigandBDBM50006019
Substrate/Competitorn/a
Meas. Tech.ChEBML_221704
IC50 9090±n/a nM
Citation Wissner, ACarroll, MLGreen, KEKerwar, SSPickett, WCSchaub, RETorley, LWWrenn, SKohler, CA Analogues of platelet activating factor. 6. Mono- and bis-aryl phosphate antagonists of platelet activating factor. J Med Chem35:1650-62 (1992) [PubMed]  Article
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Platelet activating factor receptor
Name:Platelet activating factor receptor
Synonyms:PAF-R | Platelet-activating factor receptor
Type:Protein
Mol. Mass.:39005.63
Organism:Cavia porcellus
Description:n/a
Residue:342
Sequence:
MELNSSSRVDSEFRYTLFPIVYSIIFVLGIIANGYVLWVFARLYPSKKLNEIKIFMVNLT
VADLLFLITLPLWIVYYSNQGNWFLPKFLCNLAGCLFFINTYCSVAFLGVITYNRFQAVK
YPIKTAQATTRKRGIALSLVIWVAIVAAASYFLVMDSTNVVSNKAGSGNITRCFEHYEKG
SKPVLIIHICIVLGFFIVFLLILFCNLVIIHTLLRQPVKQQRNAEVRRRALWMVCTVLAV
FVICFVPHHMVQLPWTLAELGMWPSSNHQAINDAHQVTLCLLSTNCVLDPVIYCFLTKKF
RKHLSEKLNIMRSSQKCSRVTTDTGTEMAIPINHTPVNPIKN
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  Blast E-value cutoff:
BDBM50006019
NameBDBM50006019
Synonyms:1-{3-[Hydroxy-(2-methoxy-3-tetradecyloxy-phenoxy)-phosphoryloxy]-benzyl}-pyridinium | CHEMBL297298
TypeSmall organic molecule
Emp. Form.C33H46NO6P
Mol. Mass.583.6952
SMILESCCCCCCCCCCCCCCOc1cccc(OP([O-])(=O)Oc2cccc(C[n+]3ccccc3)c2)c1OC
Structure
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n/a