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TargetLTB4R
LigandBDBM50042153
Substrate/Competitorn/a
Meas. Tech.ChEMBL_99839
Ki 3±n/a nM
Citation Kingsbury, WDPendrak, ILeber, JDBoehm, JCMallet, BSarau, HMFoley, JJSchmidt, DBDaines, RA Synthesis of structural analogs of leukotriene B4 and their receptor binding activity. J Med Chem36:3308-20 (1993) [PubMed]
More Info.:Get all data from this article,  Assay Method
 
LTB4R
Name:LTB4R
Synonyms:Chemoattractant receptor-like 1 | G-protein coupled receptor 16 | LTB4-R 1 | Leukotriene B4 R1 | Leukotriene B4 receptor | Leukotriene B4 receptor 1 | P2Y purinoceptor 7 | P2Y7
Type:Enzyme Catalytic Domain
Mol. Mass.:37582.68
Organism:HUMAN
Description:Leukotriene B4 R1 LTB4R HUMAN::Q15722
Residue:352
Sequence:
MNTTSSAAPPSLGVEFISLLAIILLSVALAVGLPGNSFVVWSILKRMQKRSVTALMVLNL
ALADLAVLLTAPFFLHFLAQGTWSFGLAGCRLCHYVCGVSMYASVLLITAMSLDRSLAVA
RPFVSQKLRTKAMARRVLAGIWVLSFLLATPVLAYRTVVPWKTNMSLCFPRYPSEGHRAF
HLIFEAVTGFLLPFLAVVASYSDIGRRLQARRFRRSRRTGRLVVLIILTFAAFWLPYHVV
NLAEAGRALAGQAAGLGLVGKRLSLARNVLIALAFLSSSVNPVLYACAGGGLLRSAGVGF
VAKLLEGTGSEASSTRRGGSLGQTARSGPAALEPGPSESLTASSPLKLNELN
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  Blast E-value cutoff:
BDBM50042153
NameBDBM50042153
Synonyms:CHEMBL113288 | Lithium; 3-(2-{7-[3-(3-butoxy-phenyl)-3-hydroxy-propenyl]-quinolin-2-yl}-1-hydroxy-ethyl)-benzoate
TypeSmall organic molecule
Emp. Form.C27H28NO5
Mol. Mass.446.5155
SMILESCCCCOc1cccc(c1)C(O)\C=C\c1cccc(CC(O)c2cccc(c2)C([O-])=O)n1
Structure
Search PDB for entries with ligand similarity:Similarity to this molecule at least:
n/a