Reaction Details Report a problem with these data
Target
2-oxoglutarate receptor 1
Ligand
BDBM50369932
Substrate
n/a
Meas. Tech.
ChEMBL_151406 (CHEMBL754752)
Ki
41±n/a nM
Citation
 Umino, T; Yoshioka, K; Saitoh, Y; Minakawa, N; Nakata, H; Matsuda, A Nucleosides and nucleotides. 200. Reinvestigation of 5'-N-ethylcarboxamidoadenosine derivatives: structure-activity relationships for P(3) purinoceptor-like proteins. J Med Chem 44:208-14 (2001) [PubMed]  Article 
Target
Name:
2-oxoglutarate receptor 1
Synonyms:
G protein-coupled receptor 80 | Gpr80 | OXGR1_RAT | Oxgr1 | P2y15
Type:
PROTEIN
Mol. Mass.:
38385.93
Organism:
Rattus norvegicus
Description:
ChEMBL_151406
Residue:
337
Sequence:
MIETLDSPANDSDFLDYITALENCTDEQISFKMQYLPVIYSIIFLVGFPGNTVAISIYVFKMRPWKSSTIIMLNLALTDLLYLTSLPFLIHYYASGENWIFGDFMCKFIRFGFHFNLYSSILFLTCFSLFRYIVIIHPMSCFSIQKTRWAVVACAGVWVISLVAVMPMTFLITSTTRTNRSACLDLTSSDDLTTIKWYNLILTATTFCLPLLIVTLCYTTIISTLTHGPRTHSCFKQKARRLTILLLLVFYVCFLPFHILRVIRIESRLLSISCSIESHIHEAYIVSRPLAALNTFGNLLLYVVVSNNFQQAFCSAVRCKAIGDLEQAKKDSCSNNP
  
Inhibitor
Name:
BDBM50369932
Synonyms:
CHEMBL608595
Type:
Small organic molecule
Emp. Form.:
C10H12N6O5
Mol. Mass.:
296.2395
SMILES:
Nc1ncnc2n(cnc12)C1O[C@@H]([C@@H](O)[C@H]1O)C(=O)NO |r|
Structure:
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