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Target
Cathepsin B
Ligand
BDBM50371946
Substrate
n/a
Meas. Tech.
ChEMBL_464363 (CHEMBL950297)
IC50
230000±n/a nM
Citation
 Hoang, VL; Li, Y; Kim, SK Cathepsin B inhibitory activities of phthalates isolated from a marine Pseudomonas strain. Bioorg Med Chem Lett 18:2083-8 (2008) [PubMed]  Article 
Target
Name:
Cathepsin B
Synonyms:
CATB_MOUSE | Ctsb
Type:
PROTEIN
Mol. Mass.:
37275.39
Organism:
Mus musculus
Description:
ChEMBL_464363
Residue:
339
Sequence:
MWWSLILLSCLLALTSAHDKPSFHPLSDDLINYINKQNTTWQAGRNFYNVDISYLKKLCGTVLGGPKLPGRVAFGEDIDLPETFDAREQWSNCPTIGQIRDQGSCGSCWAFGAVEAISDRTCIHTNGRVNVEVSAEDLLTCCGIQCGDGCNGGYPSGAWSFWTKKGLVSGGVYNSHVGCLPYTIPPCEHHVNGSRPPCTGEGDTPRCNKSCEAGYSPSYKEDKHFGYTSYSVSNSVKEIMAEIYKNGPVEGAFTVFSDFLTYKSGVYKHEAGDMMGGHAIRILGWGVENGVPYWLAANSWNLDWGDNGFFKILRGENHCGIESEIVAGIPRTDQYWGRF
  
Inhibitor
Name:
BDBM50371946
Synonyms:
CHEMBL272485
Type:
Small organic molecule
Emp. Form.:
C16H22O4
Mol. Mass.:
278.3435
SMILES:
CCCCOC(=O)c1ccccc1C(=O)OCCCC
Structure:
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