Reaction Details Report a problem with these data
Target
Multifunctional protein ADE2
Ligand
BDBM50247809
Substrate
n/a
Meas. Tech.
ChEMBL_495249 (CHEMBL1003655)
Ki
62000±n/a nM
Citation
Firestine, SM; Wu, W; Youn, H; Davisson, VJ Interrogating the mechanism of a tight binding inhibitor of AIR carboxylase. Bioorg Med Chem 17:794-803 (2009) [PubMed] Article
More Info.:
Target
Name:
Multifunctional protein ADE2
Synonyms:
AIRC | PUR6_CHICK
Type:
PROTEIN
Mol. Mass.:
47244.84
Organism:
Gallus gallus
Description:
ChEMBL_495249
Residue:
426
Sequence:
MAPAASELKLGKKVNEGKTKEVYELPDIPGCVLMQSKDQITAGNAARKDRMEGKAAISNTTTSCVFQLLQEAGIKTAFVRKQSDTAFIAAHCEMIPIEWVCRRIATGSFLKRNPGVKEGYKFYPPKIEMFYKDDANNDPQWSEEQLIEAKFSFAGLTIGKTEVDIMARSTQAIFEILEKSWQPQNCTLVDLKIEFGVNILTKEIVLADVIDNDSWRLWPSGDRSQQKDKQSYRDLKEVTPEALQMVKRNFEWVAERVELLLKTKSQGRVVVLMGSTSDLGHCEKIKKACATFGIPCELRVTSAHKGPDETLRIKAEYEGDGIPTVFVAVAGRSNGLGPVMSGNTAYPVVNCPPLSSDWGAQDVWSSLRLPSGLGCPTTLSPEGAAQFAAQIFGLNNHLVWAKLRSNMLNTWISLKQADKKLRECTL