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Target
Solute carrier organic anion transporter family member 2A1
Ligand
BDBM50318491
Substrate
n/a
Meas. Tech.
ChEMBL_836140 (CHEMBL2077576)
Ki
286±n/a nM
Citation
 Itoh, S; Lu, R; Bao, Y; Morrow, JD; Roberts, LJ; Schuster, VL Structural determinants of substrates for the prostaglandin transporter PGT. Mol Pharmacol 50:738-42 (1996) [PubMed] 
Target
Name:
Solute carrier organic anion transporter family member 2A1
Synonyms:
Matr1 | Matrin F/G 1 | Prostaglandin transporter (PGT) | SO2A1_RAT | Slc21a2 | Slco2a1 | Solute carrier family 21 member 2
Type:
Protein
Mol. Mass.:
70404.97
Organism:
Rattus norvegicus (Rat)
Description:
Q00910
Residue:
644
Sequence:
MGLLLKPGARQGSGTSSVPDRRCPRSVFSNIKVFVLCHGLLQLCQLLYSAYFKSSLTTIEKRFGLSSSSSGLISSLNEISNATLIIFISYFGSRVNRPRMIGIGGLLLAAGAFVLTLPHFLSEPYQYTSTTDGNRSSFQTDLCQKHFGALPPSKCHSTVPDTHKETSSLWGLMVVAQLLAGIGTVPIQPFGISYVDDFAEPTNSPLYISILFAIAVFGPAFGYLLGSVMLRIFVDYGRVDTATVNLSPGDPRWIGAWWLGLLISSGFLIVTSLPFFFFPRAMSRGAERSVTAEETMQTEEDKSRGSLMDFIKRFPRIFLRLLMNPLFMLVVLSQCTFSSVIAGLSTFLNKFLEKQYGATAAYANFLIGAVNLPAAALGMLFGGILMKRFVFPLQTIPRVAATIITISMILCVPLFFMGCSTSAVAEVYPPSTSSSIHPQQPPACRRDCSCPDSFFHPVCGDNGVEYVSPCHAGCSSTNTSSEASKEPIYLNCSCVSGGSASAKTGSCPTSCAQLLLPSIFLISFAALIACISHNPLYMMVLRVVNQDEKSFAIGVQFLLMRLLAWLPAPSLYGLLIDSSCVRWNYLCSGRRGACAYYDNDALRNRYLGLQMVYKALGTLLLFFISWRMKKNREYSLQENTSGLI
  
Inhibitor
Name:
BDBM50318491
Synonyms:
7-((1R,2S)-2-((S)-3-hydroxyoct-1-enyl)-5-oxocyclopent-3-enyl)heptanoic acid | CHEMBL1084644
Type:
Small organic molecule
Emp. Form.:
C20H32O4
Mol. Mass.:
336.4657
SMILES:
CCCCC[C@H](O)C=C[C@H]1C=CC(=O)[C@@H]1CCCCCCC(O)=O |r,c:10|
Structure:
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