Reaction Details Report a problem with these data
Target
Platelet glycoprotein 4
Ligand
BDBM50395029
Substrate
n/a
Meas. Tech.
ChEMBL_858884 (CHEMBL2167930)
IC50
>10000±n/a nM
Citation
 Proulx, C; Picard, É; Boeglin, D; Pohankova, P; Chemtob, S; Ong, H; Lubell, WD Azapeptide analogues of the growth hormone releasing peptide 6 as cluster of differentiation 36 receptor ligands with reduced affinity for the growth hormone secretagogue receptor 1a. J Med Chem 55:6502-11 (2012) [PubMed]  Article 
Target
Name:
Platelet glycoprotein 4
Synonyms:
Adipocyte membrane protein | CD36_RAT | CD_antigen=CD36 | Cd36 | Fat | Fatty acid translocase | Fatty acid transport protein | GPIIIB | GPIV | Glycoprotein IIIb | PAS IV | PAS-4 | Platelet glycoprotein IV
Type:
PROTEIN
Mol. Mass.:
52740.95
Organism:
Rattus norvegicus
Description:
ChEMBL_858884
Residue:
472
Sequence:
MGCDRNCGLITGAVIGAVLAVFGGILMPVGDLLIEKTIKREVVLEEGTIAFKNWVKTGTTVYRQFWIFDVQNPEEVAKNSSKIKVKQRGPYTYRVRYLAKENITQDPKDSTVSFVQPNGAIFEPSLSVGTENDNFTVLNLAVAAAPHIYTNSFVQGVLNSLIKKSKSSMFQTRSLKELLWGYKDPFLSLVPYPISTTVGVFYPYNNTVDGVYKVFNGKDNISKVAIIDTYKGKRNLSYWESYCDMINGTDAASFPPFVEKSQTLRFFSSDICRSIYAVFESEVNLKGIPVYRFVLPANAFASPLQNPDNHCFCTEKVISNNCTSYGVLDIGKCKEGKPVYISLPHFLHASPDVSEPIEGLNPNEDEHRTYLDVEPITGFTLQFAKRLQVNILVKPARKIEALKNLKRPYIVPILWLNETGTIGDEKAEMFRNQVTGKIKLLGLVEMVLLGVGVVMFVAFMISYCACRSKNGK
  
Inhibitor
Name:
BDBM50395029
Synonyms:
CHEMBL2163439 | US9708370, CP-1A(i)
Type:
Small organic molecule
Emp. Form.:
C40H47N11O6
Mol. Mass.:
777.8713
SMILES:
C[C@H](NC(=O)[C@@H](Cc1ccccc1)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@H](C)NC(=O)N(Cc1ccccc1)NC(=O)[C@@H](N)Cc1cnc[nH]1)C(N)=O |r|
Structure:
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