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Target
Glucagon-like peptide 2 receptor
Ligand
BDBM50398385
Substrate
n/a
Meas. Tech.
ChEMBL_876141 (CHEMBL2183535)
EC50
31±n/a nM
Citation
 Yamazaki, K; Terauchi, H; Iida, D; Fukumoto, H; Suzuki, S; Kagaya, T; Aoki, M; Koyama, K; Seiki, T; Takase, K; Watanabe, M; Arai, T; Tsukahara, K; Nagakawa, J Ago-allosteric modulators of human glucagon-like peptide 2 receptor. Bioorg Med Chem Lett 22:6126-35 (2012) [PubMed]  Article 
Target
Name:
Glucagon-like peptide 2 receptor
Synonyms:
GLP-2 receptor | GLP-2-R | GLP-2R | GLP2R | GLP2R_HUMAN
Type:
PROTEIN
Mol. Mass.:
63023.90
Organism:
Homo sapiens (Human)
Description:
ChEMBL_876141
Residue:
553
Sequence:
MKLGSSRAGPGRGSAGLLPGVHELPMGIPAPWGTSPLSFHRKCSLWAPGRPFLTLVLLVSIKQVTGSLLEETTRKWAQYKQACLRDLLKEPSGIFCNGTFDQYVCWPHSSPGNVSVPCPSYLPWWSEESSGRAYRHCLAQGTWQTIENATDIWQDDSECSENHSFKQNVDRYALLSTLQLMYTVGYSFSLISLFLALTLLLFLRKLHCTRNYIHMNLFASFILRTLAVLVKDVVFYNSYSKRPDNENGWMSYLSEMSTSCRSVQVLLHYFVGANYLWLLVEGLYLHTLLEPTVLPERRLWPRYLLLGWAFPVLFVVPWGFARAHLENTGCWTTNGNKKIWWIIRGPMMLCVTVNFFIFLKILKLLISKLKAHQMCFRDYKYRLAKSTLVLIPLLGVHEILFSFITDDQVEGFAKLIRLFIQLTLSSFHGFLVALQYGFANGEVKAELRKYWVRFLLARHSGCRACVLGKDFRFLGKCPKKLSEGDGAEKLRKLQPSLNSGRLLHLAMRGLGELGAQPQQDHARWPRGSSLSECSEGDVTMANTMEEILEESEI
  
Inhibitor
Name:
BDBM50398385
Synonyms:
CHEMBL2177394
Type:
Small organic molecule
Emp. Form.:
C156H242N40O53S
Mol. Mass.:
3557.892
SMILES:
n/a
Structure:
Search PDB for entries with ligand similarity: