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Target
5-hydroxytryptamine receptor 1D
Ligand
BDBM50406752
Substrate
n/a
Meas. Tech.
ChEBML_1965
IC50
16±n/a nM
Citation
 Street, LJ; Baker, R; Castro, JL; Chambers, MS; Guiblin, AR; Hobbs, SC; Matassa, VG; Reeve, AJ; Beer, MS; Middlemiss, DN Synthesis and serotonergic activity of 5-(oxadiazolyl)tryptamines: potent agonists for 5-HT1D receptors. J Med Chem 36:1529-38 (1993) [PubMed]  Article 
Target
Name:
5-hydroxytryptamine receptor 1D
Synonyms:
5HT1D_PIG | HTR1D | Serotonin 1d (5-HT1d) receptor
Type:
PROTEIN
Mol. Mass.:
32680.56
Organism:
Sus scrofa
Description:
ChEMBL_1963
Residue:
291
Sequence:
AMTDLLVSILVMPISIPYTITQTWSFGQLLCDIWLSSDITCCTASILHLCVIALDRYWAITDALEYSKRRTAGHAAAMIAIVWAISICISIPPLFWRQARAHEEISDCLVNTSQISYTIYSTCGAFYIPSLLLIILYGRIYRAARNRILNPPSLYGKRFTTAHLITGSAGSSLCSLNPSLHEGHSHSAGSPLFFNHVKIKLADSVLERKRISAARERKATKTLGIILGAFIICWLPFFVASLVLPICRDSCWIHPALFDFFTWLGYLNSLINPIIYTVFNEEFRQAFQKVV
  
Inhibitor
Name:
BDBM50406752
Synonyms:
CHEMBL290080
Type:
Small organic molecule
Emp. Form.:
C20H20N4O2
Mol. Mass.:
348.3984
SMILES:
COc1ccccc1Cc1noc(n1)-c1ccc2[nH]cc(CCN)c2c1
Structure:
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