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Target
Melanocortin receptor 3
Ligand
BDBM50410257
Substrate
n/a
Meas. Tech.
ChEMBL_307551 (CHEMBL831264)
IC50
3162±n/a nM
Citation
Kruijtzer, JA; Nijenhuis, WA; Wanders, N; Gispen, WH; Liskamp, RM; Adan, RA Peptoid-peptide hybrids as potent novel melanocortin receptor ligands. J Med Chem 48:4224-30 (2005) [PubMed] Article
More Info.:
Target
Name:
Melanocortin receptor 3
Synonyms:
MC3-R | MC3R | MC3R_HUMAN | Melanocortin MC3 | Melanocortin receptor (M3 and M4)
Type:
Enzyme
Mol. Mass.:
36044.86
Organism:
Homo sapiens (Human)
Description:
P41968
Residue:
323
Sequence:
MNASCCLPSVQPTLPNGSEHLQAPFFSNQSSSAFCEQVFIKPEVFLSLGIVSLLENILVILAVVRNGNLHSPMYFFLCSLAVADMLVSVSNALETIMIAIVHSDYLTFEDQFIQHMDNIFDSMICISLVASICNLLAIAVDRYVTIFYALRYHSIMTVRKALTLIVAIWVCCGVCGVVFIVYSESKMVIVCLITMFFAMMLLMGTLYVHMFLFARLHVKRIAALPPADGVAPQQHSCMKGAVTITILLGVFIFCWAPFFLHLVLIITCPTNPYCICYTAHFNTYLVLIMCNSVIDPLIYAFRSLELRNTFREILCGCNGMNLG