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Target
Solute carrier organic anion transporter family member 2A1
Ligand
BDBM50366413
Substrate
n/a
Meas. Tech.
ChEMBL_838709 (CHEMBL2078491)
Ki
13000000±n/a nM
Citation
 Chan, BS; Endo, S; Kanai, N; Schuster, VL Identification of lactate as a driving force for prostanoid transport by prostaglandin transporter PGT. Am J Physiol Renal Physiol 282:1097-102 (2002) [PubMed]  Article 
Target
Name:
Solute carrier organic anion transporter family member 2A1
Synonyms:
OATP2A1 | Prostaglandin Transporter | SLC21A2 | SLCO2A1 | SO2A1_HUMAN
Type:
Enzyme Catalytic Domain
Mol. Mass.:
70068.67
Organism:
Homo sapiens (Human)
Description:
Prostaglandin Transporter 0 HUMAN::Q92959
Residue:
643
Sequence:
MGLLPKLGASQGSDTSTSRAGRCARSVFGNIKVFVLCQGLLQLCQLLYSAYFKSSLTTIEKRFGLSSSSSGLISSLNEISNAILIIFVSYFGSRVHRPRLIGIGGLFLAAGAFILTLPHFLSEPYQYTLASTGNNSRLQAELCQKHWQDLPPSKCHSTTQNPQKETSSMWGLMVVAQLLAGIGTVPIQPFGISYVDDFSEPSNSPLYISILFAISVFGPAFGYLLGSVMLQIFVDYGRVNTAAVNLVPGDPRWIGAWWLGLLISSALLVLTSFPFFFFPRAMPIGAKRAPATADEARKLEEAKSRGSLVDFIKRFPCIFLRLLMNSLFVLVVLAQCTFSSVIAGLSTFLNKFLEKQYGTSAAYANFLIGAVNLPAAALGMLFGGILMKRFVFSLQAIPRIATTIITISMILCVPLFFMGCSTPTVAEVYPPSTSSSIHPQSPACRRDCSCPDSIFHPVCGDNGIEYLSPCHAGCSNINMSSATSKQLIYLNCSCVTGGSASAKTGSCPVPCAHFLLPAIFLISFVSLIACISHNPLYMMVLRVVNQEEKSFAIGVQFLLMRLLAWLPSPALYGLTIDHSCIRWNSLCLGRRGACAYYDNDALRDRYLGLQMGYKALGMLLLCFISWRVKKNKEYNVQKAAGLI
  
Inhibitor
Name:
BDBM50366413
Synonyms:
PHOSPHOENOLPYRUVATE
Type:
Small organic molecule
Emp. Form.:
C3H5O6P
Mol. Mass.:
168.042
SMILES:
OC(=O)C(=C)OP(O)(O)=O
Structure:
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