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TargetAdrenaline alpha1
LigandBDBM50367247
Substrate/Competitorn/a
Meas. Tech.ChEMBL_838515
Ki 4300±n/a nM
Citation Martel, FVetter, TRuss, HGründemann, DAzevedo, IKoepsell, HSchömig, E Transport of small organic cations in the rat liver. The role of the organic cation transporter OCT1. Naunyn Schmiedebergs Arch Pharmacol354:320-6 (1997) [PubMed]
More Info.:Get all data from this article,  Assay Method
 
Adrenaline alpha1
Name:Adrenaline alpha1
Synonyms:Oct1 | Organic cation transporter 1 | Slc22a1 | Solute carrier family 22 member 1 | adrenergic Alpha1 | rOCT1
Type:Enzyme Catalytic Domain
Mol. Mass.:61538.40
Organism:RAT
Description:Adrenaline alpha1 0 RAT::Q63089
Residue:556
Sequence:
MPTVDDVLEQVGEFGWFQKQAFLLLCLISASLAPIYVGIVFLGFTPGHYCQNPGVAELSQ
RCGWSQAEELNYTVPGLGPSDEASFLSQCMRYEVDWNQSTLDCVDPLSSLVANRSQLPLG
PCEHGWVYDTPGSSIVTEFNLVCGDAWKVDLFQSCVNLGFFLGSLVVGYIADRFGRKLCL
LVTTLVTSVSGVLTAVAPDYTSMLLFRLLQGMVSKGSWVSGYTLITEFVGSGYRRTTAIL
YQMAFTVGLVGLAGVAYAIPDWRWLQLAVSLPTFLFLLYYWFVPESPRWLLSQKRTTRAV
RIMEQIAQKNGKVPPADLKMLCLEEDASEKRSPSFADLFRTPNLRKHTVILMYLWFSCAV
LYQGLIMHVGATGANLYLDFFYSSLVEFPAAFIILVTIDRIGRIYPIAASNLVTGAACLL
MIFIPHELHWLNVTLACLGRMGATIVLQMVCLVNAELYPTFIRNLGMMVCSALCDLGGIF
TPFMVFRLMEVWQALPLILFGVLGLTAGAMTLLLPETKGVALPETIEEAENLGRRKSKAK
ENTIYLQVQTGKSSST
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BDBM50367247
NameBDBM50367247
Synonyms:QUININE | Quinamm | Quinsan | cid_3034034
TypeSmall organic molecule
Emp. Form.C20H24N2O2
Mol. Mass.324.4168
SMILESCOc1ccc2nccc([C@@H](O)[C@@H]3C[C@@H]4CCN3C[C@@H]4C=C)c2c1 |THB:20:19:12.13:16.15,10:12:19.18:16.15|
Structure
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