Reaction Details Report a problem with these data
Target
Lysophosphatidic acid receptor 5
Ligand
BDBM50148348
Substrate
n/a
Meas. Tech.
ChEMBL_946256 (CHEMBL2344994)
EC50
55±n/a nM
Citation
 Jiang, G; Inoue, A; Aoki, J; Prestwich, GD Phosphorothioate analogs of sn-2 radyl lysophosphatidic acid (LPA): metabolically stabilized LPA receptor agonists. Bioorg Med Chem Lett 23:1865-9 (2013) [PubMed]  Article 
Target
Name:
Lysophosphatidic acid receptor 5
Synonyms:
GPR92 | GPR93 | LPAR5 | LPAR5_HUMAN | Lysophosphatidic acid receptor 5 | Lysophosphatidic acid receptor 5 (LPA5)
Type:
Enzyme
Mol. Mass.:
41372.36
Organism:
Homo sapiens (Human)
Description:
Q9H1C0
Residue:
372
Sequence:
MLANSSSTNSSVLPCPDYRPTHRLHLVVYSLVLAAGLPLNALALWVFLRALRVHSVVSVYMCNLAASDLLFTLSLPVRLSYYALHHWPFPDLLCQTTGAIFQMNMYGSCIFLMLINVDRYAAIVHPLRLRHLRRPRVARLLCLGVWALILVFAVPAARVHRPSRCRYRDLEVRLCFESFSDELWKGRLLPLVLLAEALGFLLPLAAVVYSSGRVFWTLARPDATQSQRRRKTVRLLLANLVIFLLCFVPYNSTLAVYGLLRSKLVAASVPARDRVRGVLMVMVLLAGANCVLDPLVYYFSAEGFRNTLRGLGTPHRARTSATNGTRAALAQSERSAVTTDATRPDAASQGLLRPSDSHSLSSFTQCPQDSAL
  
Inhibitor
Name:
BDBM50148348
Synonyms:
(R)-Octadec-9-enoic acid 2-hydroxy-3-phosphonooxy-propyl ester | 1-oleoyl lysophosphatidic acid | CHEMBL117021 | lysophosphatidic acid
Type:
Small organic molecule
Emp. Form.:
C21H41O7P
Mol. Mass.:
436.5198
SMILES:
CCCCCCCC\C=C/CCCCCCCC(=O)OC[C@@H](O)COP(O)(O)=O
Structure:
Search PDB for entries with ligand similarity: