Reaction Details Report a problem with these data
Target
P2Y purinoceptor 11
Ligand
BDBM50435011
Substrate
n/a
Meas. Tech.
ChEMBL_963120 (CHEMBL2390599)
EC50
3680±n/a nM
Citation
Azran, S; Förster, D; Danino, O; Nadel, Y; Reiser, G; Fischer, B Highly efficient biocompatible neuroprotectants with dual activity as antioxidants and P2Y receptor agonists. J Med Chem 56:4938-52 (2013) [PubMed] Article
More Info.:
Target
Name:
P2Y purinoceptor 11
Synonyms:
P2RY11 | P2Y purinoceptor 11 | P2Y11 | P2Y11_HUMAN | Purinergic receptor P2Y11
Type:
PROTEIN
Mol. Mass.:
40366.02
Organism:
Homo sapiens (Human)
Description:
ChEMBL_1362532
Residue:
374
Sequence:
MAANVSGAKSCPANFLAAADDKLSGFQGDFLWPILVVEFLVAVASNGLALYRFSIRKQRPWHPAVVFSVQLAVSDLLCALTLPPLAAYLYPPKHWRYGEAACRLERFLFTCNLLGSVIFITCISLNRYLGIVHPFFARSHLRPKHAWAVSAAGWVLAALLAMPTLSFSHLKRPQQGAGNCSVARPEACIKCLGTADHGLAAYRAYSLVLAGLGCGLPLLLTLAAYGALGRAVLRSPGMTVAEKLRVAALVASGVALYASSYVPYHIMRVLNVDARRRWSTRCPSFADIAQATAALELGPYVGYQVMRGLMPLAFCVHPLLYMAAVPSLGCCCRHCPGYRDSWNPEDAKSTGQALPLNATAAPKPSEPQSRELSQ