Reaction Details Report a problem with these data
Target
C-C chemokine receptor type 1
Ligand
BDBM50436256
Substrate
n/a
Meas. Tech.
ChEMBL_966430 (CHEMBL2398867)
IC50
1.000000±n/a nM
Citation
Gardner, DS; Santella, JB; Duncia, JV; Carter, PH; Dhar, TG; Wu, H; Guo, W; Cavallaro, C; Van Kirk, K; Yarde, M; Briceno, SW; Grafstrom, RR; Liu, R; Patel, SR; Tebben, AJ; Camac, D; Khan, J; Watson, A; Yang, G; Rose, A; Foster, WR; Cvijic, ME; Davies, P; Hynes, J The discovery of BMS-457, a potent and selective CCR1 antagonist. Bioorg Med Chem Lett 23:3833-40 (2013) [PubMed] Article
More Info.:
Target
Name:
C-C chemokine receptor type 1
Synonyms:
C-C CKR-1 | C-C chemokine receptor type 1 (CCR1) | CC-CKR-1 | CCR-1 | CCR1 | CCR1_HUMAN | CD_antigen=CD191 | CMKBR1 | CMKR1 | HM145 | LD78 receptor | MIP-1alpha-R | Macrophage inflammatory protein 1-alpha receptor | RANTES-R | SCYAR1
Type:
Enzyme
Mol. Mass.:
41180.69
Organism:
Homo sapiens (Human)
Description:
P32246
Residue:
355
Sequence:
METPNTTEDYDTTTEFDYGDATPCQKVNERAFGAQLLPPLYSLVFVIGLVGNILVVLVLVQYKRLKNMTSIYLLNLAISDLLFLFTLPFWIDYKLKDDWVFGDAMCKILSGFYYTGLYSEIFFIILLTIDRYLAIVHAVFALRARTVTFGVITSIIIWALAILASMPGLYFSKTQWEFTHHTCSLHFPHESLREWKLFQALKLNLFGLVLPLLVMIICYTGIIKILLRRPNEKKSKAVRLIFVIMIIFFLFWTPYNLTILISVFQDFLFTHECEQSRHLDLAVQVTEVIAYTHCCVNPVIYAFVGERFRKYLRQLFHRRVAVHLVKWLPFLSVDRLERVSSTSPSTGEHELSAGF