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Target
G-protein coupled receptor 35
Ligand
BDBM50440040
Substrate
n/a
Meas. Tech.
ChEMBL_982932 (CHEMBL2429572)
EC50
5.5±n/a nM
Citation
 Thimm, D; Funke, M; Meyer, A; Müller, CE 6-Bromo-8-(4-[(3)H]methoxybenzamido)-4-oxo-4H-chromene-2-carboxylic Acid: a powerful tool for studying orphan G protein-coupled receptor GPR35. J Med Chem 56:7084-99 (2013) [PubMed]  Article 
Target
Name:
G-protein coupled receptor 35
Synonyms:
G protein-coupled receptor 35 | GPR35 | GPR35_HUMAN
Type:
Enzyme Catalytic Domain
Mol. Mass.:
34085.57
Organism:
Homo sapiens (Human)
Description:
gi_33695097
Residue:
309
Sequence:
MNGTYNTCGSSDLTWPPAIKLGFYAYLGVLLVLGLLLNSLALWVFCCRMQQWTETRIYMTNLAVADLCLLCTLPFVLHSLRDTSDTPLCQLSQGIYLTNRYMSISLVTAIAVDRYVAVRHPLRARGLRSPRQAAAVCAVLWVLVIGSLVARWLLGIQEGGFCFRSTRHNFNSMAFPLLGFYLPLAVVVFCSLKVVTALAQRPPTDVGQAEATRKAARMVWANLLVFVVCFLPLHVGLTVRLAVGWNACALLETIRRALYITSKLSDANCCLDAICYYYMAKEFQEASALAVAPSAKAHKSQDSLCVTLA
  
Inhibitor
Name:
BDBM50440040
Synonyms:
CHEMBL2425821
Type:
Small organic molecule
Emp. Form.:
C18H10BrF2NO6
Mol. Mass.:
454.176
SMILES:
COc1cc(F)c(C(=O)Nc2cc(Br)cc3c2oc(cc3=O)C(O)=O)c(F)c1
Structure:
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