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Target
Beta-2 adrenergic receptor
Ligand
BDBM50421732
Substrate
n/a
Meas. Tech.
ChEBML_37819
Kd
6470±n/a nM
Citation
 IJzerman, AP; Bultsma, T; Timmerman, H Quantitative evaluation of the beta 2-adrenoceptor intrinsic activity of N-tert-butylphenylethanolamines. J Med Chem 29:549-54 (1986) [PubMed]  Article 
Target
Name:
Beta-2 adrenergic receptor
Synonyms:
ADRB2 | ADRB2_BOVIN | Beta-2 adrenergic receptor | Beta-2 adrenoceptor | Beta-2 adrenoreceptor | adrenergic Beta
Type:
Enzyme Catalytic Domain
Mol. Mass.:
47141.18
Organism:
BOVINE
Description:
adrenergic Beta ADRB2 BOVINE::Q28044
Residue:
418
Sequence:
MGQPGNRSVFLLAPNASHAPDQNVTLERDEAWVVGMGILMSLIVLAIVFGNVLVITAIAKFERLQTVTNYFITSLACADLVMGLAVVPFGACHILMKMWTFGNFWCEFWTSIDVLCVTASIETLCVIAVDRYLAITSPFKYQCLLTKNKARVVILMVWIVSGLTSFLPIQMHWYRASHKEAINCYAKETCCDFFTNQPYAIASSIVSFYLPLVVMVFVYSRVFQVAKRQLQKIDKSEGRFHAQNVSQVEQDGRSGLGQRRTSKFYLKEHKALKTLGIIMGTFTLCWLPFFIVNIVHVIKDNLIRKEIYILLNWLGYINSAFNPLIYCRSPDFRIAFQELLCLRRSSLKAYGNGCSSNSNDRTDYTGEQSGYHLGEEKDSELLCEDPPGTENFVNQQGTVPSDSIDSQGRNCSTNDSLL
  
Inhibitor
Name:
BDBM50421732
Synonyms:
CHEMBL1159711 | VUF8303
Type:
Small organic molecule
Emp. Form.:
C12H17Cl2NO2
Mol. Mass.:
278.175
SMILES:
CC(C)(C)NCC(O)c1cc(Cl)c(O)c(Cl)c1
Structure:
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