Reaction Details Report a problem with these data
Target
Chromobox protein homolog 8
Ligand
BDBM50009555
Substrate
n/a
Meas. Tech.
ChEMBL_1336413 (CHEMBL3242417)
Kd
1890±n/a nM
Citation
Simhadri, C; Daze, KD; Douglas, SF; Quon, TT; Dev, A; Gignac, MC; Peng, F; Heller, M; Boulanger, MJ; Wulff, JE; Hof, F Chromodomain antagonists that target the polycomb-group methyllysine reader protein chromobox homolog 7 (CBX7). J Med Chem 57:2874-83 (2014) [PubMed] Article
More Info.:
Target
Name:
Chromobox protein homolog 8
Synonyms:
CBX8 | CBX8_HUMAN | PC3 | Polycomb 3 homolog | RC1 | Rectachrome 1 | hPc3
Type:
PROTEIN
Mol. Mass.:
43415.86
Organism:
Homo sapiens (Human)
Description:
ChEMBL_108272
Residue:
389
Sequence:
MELSAVGERVFAAEALLKRRIRKGRMEYLVKWKGWSQKYSTWEPEENILDARLLAAFEEREREMELYGPKKRGPKPKTFLLKAQAKAKAKTYEFRSDSARGIRIPYPGRSPQDLASTSRAREGLRNMGLSPPASSTSTSSTCRAEAPRDRDRDRDRDRERDRERERERERERERERERERGTSRVDDKPSSPGDSSKKRGPKPRKELPDPSQRPLGEPSAGLGEYLKGRKLDDTPSGAGKFPAGHSVIQLARRQDSDLVQCGVTSPSSAEATGKLAVDTFPARVIKHRAAFLEAKGQGALDPNGTRVRHGSGPPSSGGGLYRDMGAQGGRPSLIARIPVARILGDPEEESWSPSLTNLEKVVVTDVTSNFLTVTIKESNTDQGFFKEKR