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Target
Casein kinase I isoform gamma-3
Ligand
BDBM50025019
Substrate
n/a
Meas. Tech.
ChEMBL_1440403 (CHEMBL3386216)
IC50
810±n/a nM
Citation
Richter, J; Bischof, J; Zaja, M; Kohlhof, H; Othersen, O; Vitt, D; Alscher, V; Pospiech, I; García-Reyes, B; Berg, S; Leban, J; Knippschild, U Difluoro-dioxolo-benzoimidazol-benzamides as potent inhibitors of CK1d ande with nanomolar inhibitory activity on cancer cell proliferation. J Med Chem 57:7933-46 (2014) [PubMed] Article
More Info.:
Target
Name:
Casein kinase I isoform gamma-3
Synonyms:
CSNK1G3 | KC1G3_HUMAN
Type:
PROTEIN
Mol. Mass.:
51411.12
Organism:
Homo sapiens (Human)
Description:
ChEMBL_1440403
Residue:
447
Sequence:
MENKKKDKDKSDDRMARPSGRSGHNTRGTGSSSSGVLMVGPNFRVGKKIGCGNFGELRLGKNLYTNEYVAIKLEPMKSRAPQLHLEYRFYKQLGSGDGIPQVYYFGPCGKYNAMVLELLGPSLEDLFDLCDRTFSLKTVLMIAIQLISRMEYVHSKNLIYRDVKPENFLIGRPGNKTQQVIHIIDFGLAKEYIDPETKKHIPYREHKSLTGTARYMSINTHLGKEQSRRDDLEALGHMFMYFLRGSLPWQGLKADTLKERYQKIGDTKRATPIEVLCENFPEMATYLRYVRRLDFFEKPDYDYLRKLFTDLFDRKGYMFDYEYDWIGKQLPTPVGAVQQDPALSSNREAHQHRDKMQQSKNQSADHRAAWDSQQANPHHLRAHLAADRHGGSVQVVSSTNGELNTDDPTAGRSNAPITAPTEVEVMDETKCCCFFKRRKRKTIQRHK