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Target
Taste receptor type 2 member 16
Ligand
BDBM50044849
Substrate
n/a
Meas. Tech.
ChEMBL_1456200 (CHEMBL3361955)
IC50
<39811±n/a nM
Citation
 Sparks, SM; Chen, G; Collins, JL; Danger, D; Dock, ST; Jayawickreme, C; Jenkinson, S; Laudeman, C; Leesnitzer, MA; Liang, X; Maloney, P; McCoy, DC; Moncol, D; Rash, V; Rimele, T; Vulimiri, P; Way, JM; Ross, S Identification of diarylsulfonamides as agonists of the free fatty acid receptor 4 (FFA4/GPR120). Bioorg Med Chem Lett 24:3100-3 (2014) [PubMed]  Article 
Target
Name:
Taste receptor type 2 member 16
Synonyms:
T2R16 | T2R16_HUMAN | TAS2R16 | Taste receptor type 2 member 16
Type:
PROTEIN
Mol. Mass.:
34001.15
Organism:
Homo sapiens (Human)
Description:
ChEMBL_109435
Residue:
291
Sequence:
MIPIQLTVFFMIIYVLESLTIIVQSSLIVAVLGREWLQVRRLMPVDMILISLGISRFCLQWASMLNNFCSYFNLNYVLCNLTITWEFFNILTFWLNSLLTVFYCIKVSSFTHHIFLWLRWRILRLFPWILLGSLMITCVTIIPSAIGNYIQIQLLTMEHLPRNSTVTDKLENFHQYQFQAHTVALVIPFILFLASTIFLMASLTKQIQHHSTGHCNPSMKARFTALRSLAVLFIVFTSYFLTILITIIGTLFDKRCWLWVWEAFVYAFILMHSTSLMLSSPTLKRILKGKC
  
Inhibitor
Name:
BDBM50044849
Synonyms:
CHEMBL3311308
Type:
Small organic molecule
Emp. Form.:
C16H19NO3S
Mol. Mass.:
305.392
SMILES:
COc1ccc(cc1)S(=O)(=O)Nc1c(C)cc(C)cc1C
Structure:
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