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TargetTG 1019
LigandBDBM50054794
Substrate/Competitorn/a
Meas. Tech.ChEMBL_1453946
IC50 2.7±n/a nM
Citation Patel, PReddy, CNGore, VChourey, SYe, QOuedraogo, YPGravel, SPowell, WSRokach, J Two Potent OXE-R Antagonists: Assignment of Stereochemistry. ACS Med Chem Lett5:815-9 (2014) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
TG 1019
Name:TG 1019
Synonyms:5-oxo-ETE G-protein coupled receptor | G-protein coupled receptor 170 | G-protein coupled receptor R527 | G-protein coupled receptor TG1019 | Oxoeicosanoid receptor 1
Type:Enzyme Catalytic Domain
Mol. Mass.:45833.20
Organism:HUMAN
Description:TG 1019 0 HUMAN::Q8TDS5
Residue:423
Sequence:
MLCHRGGQLIVPIIPLCPEHSCRGRRLQNLLSGPWPKQPMELHNLSSPSPSLSSSVLPPS
FSPSPSSAPSAFTTVGGSSGGPCHPTSSSLVSAFLAPILALEFVLGLVGNSLALFIFCIH
TRPWTSNTVFLVSLVAADFLLISNLPLRVDYYLLHETWRFGAAACKVNLFMLSTNRTASV
VFLTAIALNRYLKVVQPHHVLSRASVGAAARVAGGLWVGILLLNGHLLLSTFSGPSCLSY
RVGTKPSASLRWHQALYLLEFFLPLALILFAIVSIGLTIRNRGLGGQAGPQRAMRVLAMV
VAVYTICFLPSIIFGMASMVAFWLSACRSLDLCTQLFHGSLAFTYLNSVLDPVLYCFSSP
NFLHQSRALLGLTRGRQGPVSDESSYQPSRQWRYREASRKAEAIGKLKVQGEVSLEKEGS
SQG
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM50054794
n/a
NameBDBM50054794
Synonyms:CHEMBL3341971
TypeSmall organic molecule
Emp. Form.C21H28ClNO3
Mol. Mass.377.905
SMILESCCCCCCc1c(C(=O)C[C@@H](C)CC(O)=O)c2cc(Cl)ccc2n1C |r|
Structure
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