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Target
Probable G-protein coupled receptor 174
Ligand
BDBM50096442
Substrate
n/a
Meas. Tech.
ChEMBL_1495910 (CHEMBL3579721)
EC50
76±n/a nM
Citation
 Ikubo, M; Inoue, A; Nakamura, S; Jung, S; Sayama, M; Otani, Y; Uwamizu, A; Suzuki, K; Kishi, T; Shuto, A; Ishiguro, J; Okudaira, M; Kano, K; Makide, K; Aoki, J; Ohwada, T Structure-activity relationships of lysophosphatidylserine analogs as agonists of G-protein-coupled receptors GPR34, P2Y10, and GPR174. J Med Chem 58:4204-19 (2015) [PubMed]  Article 
Target
Name:
Probable G-protein coupled receptor 174
Synonyms:
GP174_HUMAN | GPCR17 | GPR174 | Probable G-protein coupled receptor 174
Type:
PROTEIN
Mol. Mass.:
38513.81
Organism:
Homo sapiens (Human)
Description:
ChEMBL_109763
Residue:
333
Sequence:
MPANYTCTRPDGDNTDFRYFIYAVTYTVILVPGLIGNILALWVFYGYMKETKRAVIFMINLAIADLLQVLSLPLRIFYYLNHDWPFGPGLCMFCFYLKYVNMYASIYFLVCISVRRFWFLMYPFRFHDCKQKYDLYISIAGWLIICLACVLFPLLRTSDDTSGNRTKCFVDLPTRNVNLAQSVVMMTIGELIGFVTPLLIVLYCTWKTVLSLQDKYPMAQDLGEKQKALKMILTCAGVFLICFAPYHFSFPLDFLVKSNEIKSCLARRVILIFHSVALCLASLNSCLDPVIYYFSTNEFRRRLSRQDLHDSIQLHAKSFVSNHTASTMTPELC
  
Inhibitor
Name:
BDBM50096442
Synonyms:
CHEMBL3577173
Type:
Small organic molecule
Emp. Form.:
C26H44NO10P
Mol. Mass.:
561.602
SMILES:
CCCCCCCCCCCOc1ccc(CCC(=O)OC[C@@H](O)COP(O)(=O)OC[C@H](N)C(O)=O)cc1 |r|
Structure:
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